A one-pot synthetic strategy for construction of the dibenzodiazepine skeleton via a transition metal-free process.

نویسندگان

  • Shuai Fang
  • Xiaoyi Niu
  • Zeyuan Zhang
  • Yan Sun
  • Xiaomeng Si
  • Cuicui Shan
  • Lei Wei
  • Aiqing Xu
  • Lei Feng
  • Chen Ma
چکیده

A one-pot transition metal-free methodology for constructing pharmacologically active dibenzodiazepine derivatives was developed. Fluoro-, bromo- and nitro-substituted aryl aldehydes were applied to this reaction efficiently.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 12 35  شماره 

صفحات  -

تاریخ انتشار 2014